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Yıl
Synthesis, characterisation and biological activity of novel 4-thiazolidinones, 1,3,4-oxadiazoles and some related compounds
SG Küçükgüzel, EE Oruç, S Rollas, F Şahin, A Özbek
European Journal of Medicinal Chemistry 37 (3), 197-206, 2002
6202002
1, 3, 4-thiadiazole derivatives. Synthesis, structure elucidation, and structure− antituberculosis activity relationship investigation
EE Oruç, S Rollas, F Kandemirli, N Shvets, AS Dimoglo
Journal of medicinal chemistry 47 (27), 6760-6767, 2004
3512004
Synthesis and characterization of novel hydrazide–hydrazones and the study of their structure–antituberculosis activity
KK Bedia, O Elçin, U Seda, K Fatma, S Nathaly, R Sevim, A Dimoglo
European journal of medicinal chemistry 41 (11), 1253-1261, 2006
3492006
Novel platinum (II) and palladium (II) complexes of thiosemicarbazones derived from 5-substitutedthiophene-2-carboxaldehydes and their antiviral and cytotoxic activities
A Karaküçük-İyidoğan, D Taşdemir, EE Oruç-Emre, J Balzarini
European journal of medicinal chemistry 46 (11), 5616-5624, 2011
1052011
Synthesis and characterization of novel hydrazide-hydrazones and the study of their structure-antituberculosis activity
B Koçyiğit-Kaymakçıoğlu, E Oruç, S Unsalan, F Kandemirli, N Shvets, ...
Eur J Med Chem 41 (11), 1253-1261, 2006
462006
New piperidine-hydrazone derivatives: Synthesis, biological evaluations and molecular docking studies as AChE and BChE inhibitors
N Karaman, Y Sıcak, T Taşkın-Tok, M Öztürk, A Karaküçük-İyidoğan, ...
European journal of medicinal chemistry 124, 270-283, 2016
442016
Antituberculosis activity of hydrazones derived from 4-fluorobenzoic acid hydrazide
B Koçyiğit-Kaymakçıoğlu, E Elçin Oruç-Emre, S Unsalan, S Rollas
Medicinal chemistry research 18, 277-286, 2009
432009
Synthesis of some novel azo derivatives of 3, 5‐dimethly‐1‐(2‐hydroxyethyl) pyrazole as potent analgesic agents
EE Oruç, B Koçyigit‐Kaymakçioglu, B Oral, HZ Altunbas‐Toklu, ...
Archiv der Pharmazie: An International Journal Pharmaceutical and Medicinal …, 2006
422006
Biting deterrence and insecticidal activity of hydrazide‐hydrazones and their corresponding 3‐acetyl‐2, 5‐disubstituted‐2, 3‐dihydro‐1, 3, 4‐oxadiazoles against Aedes aegypti
N Tabanca, A Ali, UR Bernier, IA Khan, B Kocyigit‐Kaymakcioglu, ...
Pest management science 69 (6), 703-708, 2013
362013
Designing heterocyclic chalcones, benzoyl/sulfonyl hydrazones: An insight into their biological activities and molecular docking study
BSK Aktar, Y Sıcak, TT Tok, EE Oruç-Emre, AŞ Yağlıoğlu, AK Iyidoğan, ...
Journal of Molecular Structure 1211, 128059, 2020
312020
In vivo metabolism of 4-fluorobenzoic acid [(5-nitro-2-furanyl) methylene] hydrazide in rats
NN Gülerman, EE Oruç, F Kartal, S Rollas
European journal of drug metabolism and pharmacokinetics 25, 103-108, 2000
302000
Synthesis of Novel Chiral Sulfonamide‐Bearing 1,2,4‐Triazole‐3‐thione Analogs Derived from D‐ and L‐Phenylalanine Esters as Potential Anti‐Influenza Agents
E Başaran, A Karaküçük‐Iyidoğan, D Schols, EE Oruç‐Emre
Chirality 28 (6), 495-513, 2016
292016
Microwave-assisted synthesis of new sulfonyl hydrazones, screening of biological activities and investigation of structure–activity relationship
N Karaman, EE Oruç-Emre, Y Sıcak, B Çatıkkaş, A Karaküçük-İyidoğan, ...
Medicinal Chemistry Research 25, 1590-1607, 2016
262016
Synthesis and biological activity of hydrazide–hydrazones and their corresponding 3-acetyl-2, 5-disubstituted-2, 3-dihydro-1, 3, 4-oxadiazoles
B Koçyiğit-Kaymakçıoğlu, EE Oruç-Emre, S Ünsalan, N Tabanca, SI Khan, ...
Medicinal Chemistry Research 21, 3499-3508, 2012
262012
Synthesis, molecular modeling, and biological evaluation of novel chiral thiosemicarbazone derivatives as potent anticancer agents
D Taşdemir, A Karaküçük‐İyidoğan, M Ulaşli, T Taşkin‐Tok, ...
Chirality 27 (2), 177-188, 2015
222015
Novel fluorine‐containing chiral hydrazide‐hydrazones: Design, synthesis, structural elucidation, antioxidant and anticholinesterase activity, and in silico studies
Y Sıcak, EE Oruç‐Emre, M Öztürk, T Taşkın‐Tok, A Karaküçük‐Iyidoğan
Chirality 31 (8), 603-615, 2019
202019
The in vivo metabolism of 5-(4-nitrophenyl)-4-phenyl-2, 4-dihydro-3H-1, 2, 4-triazole-3-thione in rats
EΕ Οruç, S Rollas, L Kabasakal, MK Uysal
Drug metabolism and drug interactions 15 (2-3), 127-140, 1999
201999
Anticonvulsant activity of 3, 5-dimethylpyrazole derivatives in animal models
B Kocyigit-Kaymakcioglu, RG Aker, K Tezcan, E Sakalli, S Ketenci, ...
Medicinal Chemistry Research 20, 607-614, 2011
182011
Studies on hydrazide-hydrazones derivatives as acetylcholinesterase inhibitors
U Abu Mohsen, B KAYMAKÇIOĞLU, E Oruc-Emre, Z Kaplancikli, S Rollas
Clinical and Experimental Health Sciences 5 (1), 2015
172015
Design and Bioevaluation of Novel Hydrazide-Hydrazones Derived from 4-Acetyl-N-Substituted Benzenesulfonamide
E Bozkurt, Y Sıcak, EE Oruç-Emre, AK Iyidoğan, M Öztürk
Russian Journal of Bioorganic Chemistry 46, 702-714, 2020
162020
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