Ameliorative and protective effects of ginger and its main constituents against natural, chemical and radiation-induced toxicities CGL Muhammad A. Alsherbiny, Wessam H. Abd-Elsalam, Shymaa A. El badawy, Ehab ... Food and Chemical Toxicology, 2018 | 60* | 2018 |
New octahydroquinazoline derivatives: synthesis and hypotensive activity OI El-Sabbagh, MA Shabaan, HH Kadry, ES Al-Din European Journal of Medicinal Chemistry 45 (11), 5390-5396, 2010 | 48 | 2010 |
Design, synthesis, and biological evaluation of new pyrimidine-5-carbonitrile derivatives bearing 1, 3-thiazole moiety as novel anti-inflammatory EGFR inhibitors with cardiac … SA Abdel-Aziz, ES Taher, P Lan, GF Asaad, HAM Gomaa, NA El-Koussi, ... Bioorganic Chemistry 111, 104890, 2021 | 44 | 2021 |
Synthesis, Antimicrobial, Anti-Virulence and Anticancer Evaluation of New 5(4H)-Oxazolone-Based Sulfonamides AJ Almalki, TS Ibrahim, ES Taher, MFA Mohamed, M Youns, ... Molecules 27 (3), 671, 2022 | 38 | 2022 |
Design, synthesis and biological evaluation of novel 5-((substituted quinolin-3-yl/1-naphthyl) methylene)-3-substituted imidazolidin-2, 4-dione as HIV-1 fusion inhibitors TS Ibrahim, RM Bokhtia, AMM Al-Mahmoudy, ES Taher, MA AlAwadh, ... Bioorganic Chemistry 99, 103782, 2020 | 35 | 2020 |
The Exploitation of Enzymatically‐Derived cis‐1,2‐Dihydrocatechols and Related Compounds in the Synthesis of Biologically Active Natural Products ES Taher, MG Banwell, JN Buckler, Q Yan, P Lan The Chemical Record 18 (2), 239-264, 2018 | 34 | 2018 |
Chemoenzymatic synthesis of (+)-asperpentyn and the enantiomer of the structure assigned to aspergillusol A P Lan, LE White, ES Taher, PE Guest, MG Banwell, AC Willis Journal of natural products 78 (8), 1963-1968, 2015 | 33 | 2015 |
Synthesis of new nonclassical acridines, quinolines, and quinazolines derived from dimedone for biological evaluation OIE Sabbagh, MA Shabaan, HH Kadry, ES Al‐Din Archiv der Pharmazie 343 (9), 519-527, 2010 | 30 | 2010 |
Chemoenzymatic total synthesis of (+)-oxycodone from phenethyl acetate MAA Endoma-Arias, M Makarova, HED Paz, T Hudlicky Synthesis 51 (01), 225-232, 2019 | 25 | 2019 |
Novel benzenesulfonamide and 1, 2-benzisothiazol-3 (2H)-one-1, 1-dioxide derivatives as potential selective COX-2 inhibitors ES Taher, TS Ibrahim, M Fares, AMM Al-Mahmoudy, AF Radwan, ... European Journal of Medicinal Chemistry 171, 372-382, 2019 | 24 | 2019 |
Discovery of novel quinoline-based analogues of combretastatin A-4 as tubulin polymerisation inhibitors with apoptosis inducing activity and potent anticancer effect TS Ibrahim, MM Hawwas, AM Malebari, ES Taher, AM Omar, ... Journal of Enzyme Inhibition and Medicinal Chemistry 36 (1), 802-818, 2021 | 18 | 2021 |
The synthesis of certain derivatives and analogues of (−)-and (+)-galanthamine and an assessment of their capacities to inhibit acetylcholine esterase JN Buckler, ES Taher, NJ Fraser, AC Willis, PD Carr, CJ Jackson, ... The Journal of Organic Chemistry 82 (15), 7869-7886, 2017 | 18 | 2017 |
Potent Quinoline-Containing Combretastatin A-4 Analogues: Design, Synthesis, Antiproliferative, and Anti-Tubulin Activity ZKASYAMME Tarek S. Ibrahim 1,2,* , Mohamed M. Hawwas 3, Azizah M. Malebari 1 ... Pharmaceuticals 13 (93), 1-23, 2020 | 17* | 2020 |
Design and synthesis of novel pyrazolo [3, 4-d] pyrimidin-4-one bearing quinoline scaffold as potent dual PDE5 inhibitors and apoptotic inducers for cancer therapy TS Ibrahim, MM Hawwas, ES Taher, NA Alhakamy, MA Alfaleh, ... Bioorganic Chemistry 105, 104352, 2020 | 14 | 2020 |
The synthesis of certain phomentrioloxin A analogues and their evaluation as herbicidal agents ES Taher, P Guest, A Benton, X Ma, MG Banwell, AC Willis, T Seiser, ... The Journal of Organic Chemistry 82 (1), 211-233, 2017 | 13 | 2017 |
Chemoenzymatic pathways for the synthesis of biologically active natural products MG Banwell, B Bolte, JN Buckler, EL Chang, P Lan, ES Taher, LV White, ... Journal and Proceedings of the Royal Society of New South Wales 149 (459/462 …, 2016 | 13 | 2016 |
Uracil as a Zn-binding bioisostere of the allergic benzenesulfonamide in the design of quinoline–uracil hybrids as anticancer carbonic anhydrase inhibitors SA El-Kalyoubi, ES Taher, TS Ibrahim, MF El-Behairy, AMM Al-Mahmoudy Pharmaceuticals 15 (5), 494, 2022 | 11 | 2022 |
Design, synthesis, biological evaluation, and computational studies of novel thiazolo-pyrazole hybrids as promising selective COX-2 inhibitors: Implementation of apoptotic … AA Marzouk, ES Taher, MSA Shaykoon, P Lan, WH Abd-Allah, ... Bioorganic Chemistry 111, 104883, 2021 | 10 | 2021 |
Schiff bases as linker in the development of quinoline-sulfonamide hybrids as selective cancer-associated carbonic anhydrase isoforms IX/XII inhibitors: A new regioisomerism tactic A El-Malah, ES Taher, A Angeli, SS Elbaramawi, Z Mahmoud, N Moustafa, ... Bioorganic Chemistry 131, 106309, 2023 | 9 | 2023 |
New pyrimidine/thiazole hybrids endowed with analgesic, anti‐inflammatory, and lower cardiotoxic activities: Design, synthesis, and COX‐2/sEH dual inhibition SA Abdel‐Aziz, ES Taher, P Lan, NA El‐Koussi, OIA Salem, HAM Gomaa, ... Archiv der Pharmazie 355 (7), 2200024, 2022 | 9 | 2022 |