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Burcu Çalışkan
Burcu Çalışkan
PhD
Verified email at gazi.edu.tr - Homepage
Title
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Cited by
Year
Synthesis, analgesic, and anti-inflammatory activities of [6-(3, 5-dimethyl-4-chloropyrazole-1-yl)-3 (2H)-pyridazinon-2-yl] acetamides
M Süküroglu, BÇ Ergün, S ünlü, MF Sahin, E Küpeli, E Yesilada, ...
Archives of pharmacal research 28, 509-517, 2005
862005
Identification of novel benzimidazole derivatives as inhibitors of leukotriene biosynthesis by virtual screening targeting 5-lipoxygenase-activating protein (FLAP)
E Banoglu, B Çalışkan, S Luderer, G Eren, Y Özkan, W Altenhofen, ...
Bioorganic & medicinal chemistry 20 (12), 3728-3741, 2012
692012
Synthesis and preliminary mechanistic evaluation of 5-(p-tolyl)-1-(quinolin-2-yl) pyrazole-3-carboxylic acid amides with potent antiproliferative activity on human cancer cell …
ŞC Pirol, B Çalışkan, İ Durmaz, R Atalay, E Banoglu
European Journal of Medicinal Chemistry 87, 140-149, 2014
672014
Synthesis, antioxidant and antimicrobial evaluation of simple aromatic esters of ferulic acid
BÇ Ergün, T Çoban, FK Onurdag, E Banoglu
Archives of Pharmacal Research 34, 1251-1261, 2011
622011
Drug discovery approaches targeting 5-lipoxygenase-activating protein (FLAP) for inhibition of cellular leukotriene biosynthesis
ZT Gür, B Çalışkan, E Banoglu
European Journal of Medicinal Chemistry 153, 34-48, 2018
612018
4, 5-Diarylisoxazol-3-carboxylic acids: A new class of leukotriene biosynthesis inhibitors potentially targeting 5-lipoxygenase-activating protein (FLAP)
E Banoglu, E Çelikoğlu, S Völker, A Olgaç, J Gerstmeier, U Garscha, ...
European Journal of Medicinal Chemistry 113, 1-10, 2016
532016
The novel benzimidazole derivative BRP‐7 inhibits leukotriene biosynthesis in vitro and in vivo by targeting 5‐lipoxygenase‐activating protein (FLAP)
C Pergola, J Gerstmeier, B Mönch, B Çalışkan, S Luderer, C Weinigel, ...
British journal of pharmacology 171 (12), 3051-3064, 2014
492014
Synthesis and evaluation of analgesic, anti-inflammatory, and anticancer activities of new pyrazole-3 (5)-carboxylic acid derivatives
B Çalışkan, A Yılmaz, I Evren, S Menevşe, O Uludag, E Banoglu
Medicinal Chemistry Research 22, 782-793, 2013
432013
BRP-187: A potent inhibitor of leukotriene biosynthesis that acts through impeding the dynamic 5-lipoxygenase/5-lipoxygenase-activating protein (FLAP) complex assembly
U Garscha, S Voelker, S Pace, J Gerstmeier, B Emini, S Liening, A Rossi, ...
Biochemical pharmacology 119, 17-26, 2016
402016
Synthesis and cellular bioactivities of novel isoxazole derivatives incorporating an arylpiperazine moiety as anticancer agents
B Çalışkan, E Sinoplu, K İbiş, E Akhan Güzelcan, R Çetin Atalay, ...
Journal of enzyme inhibition and medicinal chemistry 33 (1), 1352-1361, 2018
382018
Stable ester and amide conjugates of some NSAIDs as analgesic and antiinflammatory compounds with improved biological activity
MO ULUDAĞ, BÇ ERGÜN, DA Alkan, N ERCAN, GY ÖZKAN, ...
Turkish Journal of Chemistry 35 (3), 427-439, 2011
352011
Pyrazol-3-propanoic acid derivatives as novel inhibitors of leukotriene biosynthesis in human neutrophils
B Çalışkan, S Luderer, Y Özkan, O Werz, E Banoglu
European journal of medicinal chemistry 46 (10), 5021-5033, 2011
342011
Synthesis of the amide derivatives of 3-[1-(3-pyridazinyl)-5-phenyl-1H-pyrazole-3-yl] propanoic acids as potential analgesic compounds
E Banoğlu, M ŞÜKÜROĞLU, BÇ ERGÜN, SN BAYTAŞ, E Aypar, M ARK
Turkish Journal of Chemistry 31 (6), 677-687, 2007
342007
Overview of recent drug discovery approaches for new generation leukotriene A4 hydrolase inhibitors
B Çalışkan, E Banoglu
Expert opinion on drug discovery 8 (1), 49-63, 2013
322013
Chromatographic separation and biological evaluation of benzimidazole derivative enantiomers as inhibitors of leukotriene biosynthesis
R Sardella, S Levent, F Ianni, B Çalişkan, J Gerstmeier, C Pergola, ...
Journal of Pharmaceutical and Biomedical Analysis 89, 88-92, 2014
312014
Screening and evaluation of antioxidant activity of some pyridazine derivatives
SS Caliskan B, Süküroğlu M, CobanTulay, Banoğlu E
Journal of enzyme inhibition and medicinal chemistry 23 (2), 225-229, 2008
28*2008
Identification of multi-target inhibitors of leukotriene and prostaglandin E2 biosynthesis by structural tuning of the FLAP inhibitor BRP-7
ZT Gür, B Çalışkan, UI Garscha, A Olgaç, US Schubert, J Gerstmeier, ...
European Journal of Medicinal Chemistry 150, 876-899, 2018
262018
Pyrazole derivatives as inhibitors of arachidonic acid-induced platelet aggregation
S Levent, B Çalışkan, M Çiftçi, Y Özkan, İ Yenicesu, H Ünver, E Banoglu
European Journal of Medicinal Chemistry 64, 42-53, 2013
262013
A highly potent TACC3 inhibitor as a novel anticancer drug candidate
O Akbulut, D Lengerli, O Saatci, E Duman, UOS Seker, A Isik, A Akyol, ...
Molecular cancer therapeutics 19 (6), 1243-1254, 2020
222020
Synthesis of amide derivatives of [6-(3, 5-dimethylpyrazol-1-yl)-3 (2H)-pyridazinone-2-yl] acetic acid and their analgesic and anti-inflammatory properties
E Banoğlu, Ç Akoğlu, S Ünlü, BÇ Ergün, E Küpeli, E Yeşilada, MF Şahin
Arzneimittelforschung 55 (09), 520-527, 2005
222005
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