Takip et
Gianluca SBARDELLA
Gianluca SBARDELLA
Dipartimento di Farmacia, Università di Salerno
unisa.it üzerinde doğrulanmış e-posta adresine sahip
Başlık
Alıntı yapanlar
Alıntı yapanlar
Yıl
Histone deacetylase inhibitor activity in royal jelly might facilitate caste switching in bees
A Spannhoff, YK Kim, NJM Raynal, V Gharibyan, MB Su, YY Zhou, J Li, ...
EMBO reports 12 (3), 238-243, 2011
2212011
Synthesis and Biochemical Evaluation of Δ2-Isoxazoline Derivatives as DNA Methyltransferase 1 Inhibitors
S Castellano, D Kuck, M Viviano, J Yoo, F López-Vallejo, P Conti, ...
Journal of medicinal chemistry 54 (21), 7663-7677, 2011
1922011
Arginine demethylation of G3BP1 promotes stress granule assembly
WC Tsai, S Gayatri, LC Reineke, G Sbardella, MT Bedford, RE Lloyd
Journal of Biological Chemistry 291 (43), 22671-22685, 2016
1742016
Epigenetic multiple ligands: mixed histone/protein methyltransferase, acetyltransferase, and class III deacetylase (sirtuin) inhibitors
A Mai, D Cheng, MT Bedford, S Valente, A Nebbioso, A Perrone, ...
Journal of medicinal chemistry 51 (7), 2279-2290, 2008
1622008
Dihydro(alkylthio)(naphthylmethyl)oxopyrimidines:  Novel Non-Nucleoside Reverse Transcriptase Inhibitors of the S-DABO Series
A Mai, M Artico, G Sbardella, S Quartarone, S Massa, AG Loi, A De Montis, ...
Journal of Medicinal Chemistry 40 (10), 1447-1454, 1997
1601997
5-Alkyl-2-(alkylthio)-6-(2,6-dihalophenylmethyl)-3,4-dihydropyrimidin-4(3H)-ones:  Novel Potent and Selective Dihydro-alkoxy-benzyl-oxopyrimidine Derivatives
A Mai, M Artico, G Sbardella, S Massa, E Novellino, G Greco, AG Loi, ...
Journal of Medicinal Chemistry 42 (4), 619-627, 1999
1591999
Small-molecule inhibitors of histone acetyltransferase activity: identification and biological properties
A Mai, D Rotili, D Tarantino, P Ornaghi, F Tosi, C Vicidomini, G Sbardella, ...
Journal of medicinal chemistry 49 (23), 6897-6907, 2006
1572006
Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2, 6-difluorophenyl) alkyl]-3, 4-dihydro-5-alkylpyrimidin-4 …
A Mai, G Sbardella, M Artico, R Ragno, S Massa, E Novellino, G Greco, ...
Journal of medicinal chemistry 44 (16), 2544-2554, 2001
1362001
Preparation and anti-HIV-1 activity of Thio Analogues of Dichydroalkoxybenzyloxopyrimidines
A Mai, M Artico, G Sbardella, S Massa, AG Loi, E Tramontano, P Scano, ...
Journal of medicinal chemistry 38 (17), 3258-3263, 1995
1351995
Identification of long chain alkylidenemalonates as novel small molecule modulators of histone acetyltransferases
G Sbardella, S Castellano, C Vicidomini, D Rotili, A Nebbioso, M Miceli, ...
Bioorganic & medicinal chemistry letters 18 (9), 2788-2792, 2008
1282008
Small molecule inhibitors of histone arginine methyltransferases: homology modeling, molecular docking, binding mode analysis, and biological evaluations
R Ragno, S Simeoni, S Castellano, C Vicidomini, A Mai, A Caroli, ...
Journal of medicinal chemistry 50 (6), 1241-1253, 2007
1262007
Nε-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart
C Colussi, J Rosati, S Straino, F Spallotta, R Berni, D Stilli, S Rossi, ...
Proceedings of the National Academy of Sciences 108 (7), 2795-2800, 2011
1212011
Constrained analogues of procaine as novel small molecule inhibitors of DNA methyltransferase-1
S Castellano, D Kuck, M Sala, E Novellino, F Lyko, G Sbardella
Journal of medicinal chemistry 51 (7), 2321-2325, 2008
1212008
Computer-aided design, synthesis, and anti-HIV-1 activity in vitro of 2-alkylamino-6-[1-(2, 6-difluorophenyl) alkyl]-3, 4-dihydro-5-alkylpyrimidin-4 (3 H)-ones as novel potent …
R Ragno, A Mai, G Sbardella, M Artico, S Massa, C Musiu, M Mura, ...
Journal of medicinal chemistry 47 (4), 928-934, 2004
1172004
p300/CBP-associated factor selectively regulates the extinction of conditioned fear
W Wei, CM Coelho, X Li, R Marek, S Yan, S Anderson, D Meyers, ...
Journal of Neuroscience 32 (35), 11930-11941, 2012
1022012
3-(4-Aroyl-1 H-pyrrol-2-yl)-N-hydroxy-2-propenamides, a new class of synthetic histone deacetylase inhibitors
S Massa, A Mai, G Sbardella, M Esposito, R Ragno, P Loidl, G Brosch
Journal of medicinal chemistry 44 (13), 2069-2072, 2001
1022001
Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases
A Mai, D Rotili, D Tarantino, A Nebbioso, S Castellano, G Sbardella, ...
Bioorganic & medicinal chemistry letters 19 (4), 1132-1135, 2009
972009
The emerging role of lysine methyltransferase SETD8 in human diseases
C Milite, A Feoli, M Viviano, D Rescigno, A Cianciulli, AL Balzano, A Mai, ...
Clinical epigenetics 8, 1-15, 2016
912016
Novel 3, 5-bis (bromohydroxybenzylidene) piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity
D Cheng, S Valente, S Castellano, G Sbardella, R Di Santo, R Costi, ...
Journal of medicinal chemistry 54 (13), 4928-4932, 2011
892011
A New Facile and Expeditious Synthesis of N-Hydroxy-N′-Phenyloctanediamjde, a Potent Inducer of Terminal Cytodifferecntiation
A Mai, M Esposito, G Sbardella, S Massa
Organic Preparations and Procedures International 33 (4), 391-394, 2001
882001
Sistem, işlemi şu anda gerçekleştiremiyor. Daha sonra yeniden deneyin.
Makaleler 1–20